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iloperidone improves amounts of diazepam by impacting hepatic/intestinal enzyme CYP3A4 metabolism. Use Caution/Check. Iloperidone is often a time-dependent CYP3A inhibitor and should cause elevated plasma amounts of drugs predominantly eradicated by CYP3A4.fedratinib will improve the level or impact of diazepam by influencing hepatic enzyme CYP2C19